Synthesis of irreversibly binding bicalutamide analogs for imaging studies
- 11 July 2005
- journal article
- research article
- Published by Elsevier in Tetrahedron Letters
- Vol. 46 (28) , 4821-4823
- https://doi.org/10.1016/j.tetlet.2005.04.143
Abstract
No abstract availableKeywords
This publication has 16 references indexed in Scilit:
- Synthesis of novel iodo derived bicalutamide analogsTetrahedron Letters, 2004
- A Ligand-Based Approach To Identify Quantitative Structure−Activity Relationships for the Androgen ReceptorJournal of Medicinal Chemistry, 2004
- Design, Synthesis, and Biological Characterization of Metabolically Stable Selective Androgen Receptor ModulatorsJournal of Medicinal Chemistry, 2004
- Pharmacodynamics of Selective Androgen Receptor ModulatorsThe Journal of Pharmacology and Experimental Therapeutics, 2003
- Pharmacology, Pharmacokinetics, and Metabolism of Acetothiolutamide, a Novel Nonsteroidal Agonist for the Androgen ReceptorThe Journal of Pharmacology and Experimental Therapeutics, 2003
- A Two-step Synthesis of the Anti-cancer Drug (R,S)-BicalutamideSynthesis, 2002
- Discovery of Nonsteroidal AndrogensBiochemical and Biophysical Research Communications, 1998
- The Intracellular Receptor and Signal Transducers and Activators of Transcription Factor Superfamilies: Novel Targets for Small-Molecule Drug DiscoveryJournal of Medicinal Chemistry, 1995
- Non-steroidal antiandrogens. Design of novel compounds based on an infrared study of the dominant conformation and hydrogen-bonding properties of a series of anilide antiandrogensJournal of Medicinal Chemistry, 1991
- Resolution of the non steroidal antiandrogen 4'-cyano-3-[(4-fluorophenyl)sulfonyl]-2-hydroxy-2-methyl-3'-(trifluoromethyl)propionanilide and the determination of the absolute configuration of the active enantiomerJournal of Medicinal Chemistry, 1988