Binding of (−)-[3H]-CGP12177 at two sites in recombinant human β1-adrenoceptors and interaction with β-blockers
- 1 May 2004
- journal article
- research article
- Published by Springer Nature in Naunyn-Schmiedebergs Archiv für experimentelle Pathologie und Pharmakologie
- Vol. 369 (5) , 525-532
- https://doi.org/10.1007/s00210-004-0884-y
Abstract
No abstract availableKeywords
This publication has 27 references indexed in Scilit:
- Comparison of the affinity of β‐blockers for two states of the β1‐adrenoceptor in ferret ventricular myocardiumBritish Journal of Pharmacology, 2002
- Putative β4‐adrenoceptors in rat ventricle mediate increases in contractile force and cell Ca2+: comparison with atrial receptors and relationship to (−)‐[3H]‐CGP 12177 bindingBritish Journal of Pharmacology, 1999
- Desensitization and resensitization of β1‐ and putative β4‐adrenoceptor mediated responses occur in parallel in a rat model of cardiac failureBritish Journal of Pharmacology, 1999
- Action potential shortening through the putative β4‐adrenoceptor in ferret ventricle: comparison with β1‐ and β2‐adrenoceptor‐mediated effectsBritish Journal of Pharmacology, 1998
- Validity of (−)‐[3H]‐CGP 12177A as a radioligand for the ‘putative β4‐adrenoceptor’ in rat atriumBritish Journal of Pharmacology, 1998
- Stimulation of cyclic AMP‐dependent protein kinase in rat atria by (–;)‐CGP 12177 through an atypical β‐adrenoceptorBritish Journal of Pharmacology, 1997
- (−)-Timolol is a more potent antagonist of the positive inotropic effects of (−)-adrenaline than of those of (−)-noradrenaline in human atriumPublished by Wiley ,1996
- Anomalous Behavior of CGP 12177A ON β2-Adrenergic ReceptorsJournal of Receptors and Signal Transduction, 1996
- Is there a third heart β-adrenoceptor?Trends in Pharmacological Sciences, 1989
- Decreased Catecholamine Sensitivity and β-Adrenergic-Receptor Density in Failing Human HeartsNew England Journal of Medicine, 1982