A designed P1 cysteine mimetic for covalent and non-covalent inhibitors of HCV NS3 protease
- 6 February 2002
- journal article
- research article
- Published by Elsevier in Bioorganic & Medicinal Chemistry Letters
- Vol. 12 (4) , 701-704
- https://doi.org/10.1016/s0960-894x(01)00842-3
Abstract
No abstract availableKeywords
This publication has 24 references indexed in Scilit:
- On the size of the active site in proteases. I. PapainPublished by Elsevier ,2005
- Evolution, synthesis and SAR of tripeptide α-ketoacid Inhibitors of the hepatitis C virus NS3/NS4A serine proteasePublished by Elsevier ,2002
- Synthesis, Structure−Activity Relationships, and Pharmacokinetic Profiles of Nonpeptidic α-Keto Heterocycles as Novel Inhibitors of Human ChymaseJournal of Medicinal Chemistry, 2001
- The identification of α-ketoamides as potent inhibitors of hepatitis c virus nS3-4a proteinaseBioorganic & Medicinal Chemistry Letters, 2001
- α-Ketoamides, α-ketoesters and α-diketones as HCV NS3 protease inhibitorsBioorganic & Medicinal Chemistry Letters, 2000
- Hepatitis C virus NS3/4A proteaseAntiviral Research, 1998
- The Cation−π InteractionChemical Reviews, 1997
- Hydrogen Bond Donor Properties of the Difluoromethyl GroupThe Journal of Organic Chemistry, 1995
- Falling out of the fold: tumorigenic mutations and p53Chemistry & Biology, 1994
- Sulphur‐aromatic interactions in proteinsFEBS Letters, 1985