2-Aminothiophene-3-carboxylates and carboxamides as adenosine A1 receptor allosteric enhancers
- 1 April 2006
- journal article
- Published by Elsevier in Bioorganic & Medicinal Chemistry
- Vol. 14 (7) , 2358-2365
- https://doi.org/10.1016/j.bmc.2005.11.018
Abstract
No abstract availableKeywords
This publication has 9 references indexed in Scilit:
- Synthesis of 2-amino-3-heteroaroylthiophenes and evaluation of their activity as potential allosteric enhancers at the human A1 receptorEuropean Journal of Medicinal Chemistry, 2004
- Allosteric Enhancers of A1 Adenosine Receptors Increase Receptor-G Protein Coupling and Counteract Guanine Nucleotide Effects on Agonist BindingMolecular Pharmacology, 2003
- 2-Amino-3-benzoylthiophene Allosteric Enhancers of A1 Adenosine Agonist Binding: New 3, 4-, and 5-ModificationsJournal of Medicinal Chemistry, 2003
- 2-Amino-3-aroyl-4,5-alkylthiophenes: Agonist Allosteric Enhancers at Human A1 Adenosine ReceptorsJournal of Medicinal Chemistry, 2001
- Synthesis and biological effects of a new series of 2-amino-3-benzoylthiophenes as allosteric enhancers of A1-adenosine receptorBioorganic & Medicinal Chemistry Letters, 2000
- Elucidation of structure-activity relationships of 2-amino-3-benzoylthiophenes: Study of their allosteric enhancing vs. antagonistic activity on adenosine A1 receptorsDrug Development Research, 2000
- Allosteric Modulation of the Adenosine A1 Receptor. Synthesis and Biological Evaluation of Novel 2-Amino-3-benzoylthiophenes as Allosteric Enhancers of Agonist BindingJournal of Medicinal Chemistry, 1999
- 2‐aminothiophenes by the gewald reactionJournal of Heterocyclic Chemistry, 1999
- Heterocyclen aus CH‐aciden Nitrilen, VIII. 2‐Amino‐thiophene aus methylenaktiven Nitrilen, Carbonylverbindungen und SchwefelEuropean Journal of Inorganic Chemistry, 1966