3-Amino-1-(3,4-dichloro-α-methyl-benzyl)-2-pyrazolin-5-one (Bay g 2821), a potent diuretic from a new substance class
- 1 March 1977
- journal article
- specialia
- Published by Springer Nature in Cellular and Molecular Life Sciences
- Vol. 33 (3) , 382-383
- https://doi.org/10.1007/bf02002840
Abstract
Chemistry, salidiuretic activity and mechanism of action of 3-amino-1-(3,4-dichloro-α-methyl-benzyl)-2-pyrazolin-5-one (Bay g 2821), a new diuretic, are described. Owing to the initial rapid onset of activity, the reserve in capacity and the additional long duration of activity, this substance represents a potent diuretic and antihypertensive agent.Keywords
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