A new access to 3,5-disubstituted piperazinones via Pd(0)-catalyzed amination
- 3 May 2003
- journal article
- research article
- Published by Elsevier in Tetrahedron Letters
- Vol. 44 (22) , 4213-4216
- https://doi.org/10.1016/s0040-4039(03)00885-2
Abstract
No abstract availableKeywords
This publication has 23 references indexed in Scilit:
- Molecular Simplification of 1,4-Diazabicyclo[4.3.0]nonan-9-ones Gives Piperazine Derivatives That Maintain High Nootropic ActivityJournal of Medicinal Chemistry, 2000
- Design, Synthesis, and Preliminary Pharmacological Evaluation of 1,4-Diazabicyclo[4.3.0]nonan-9-ones as a New Class of Highly Potent Nootropic AgentsJournal of Medicinal Chemistry, 2000
- Synthesis of piperazine derivatives and evaluation of their antihistamine and antibradykinin effectsBioorganic & Medicinal Chemistry Letters, 1999
- Sequential mono-N-arylation of piperazine nitrogens. Part 1: A simplified method and its application to the preparation of a key N,N′-biaryl piperazine antifungal intermediateTetrahedron Letters, 1999
- Design and synthesis of thrombin receptor-derived nonpeptide mimetics utilizing a piperazine scaffoldBioorganic & Medicinal Chemistry, 1999
- Hybridized and isosteric analogues of N 1 -acetyl- N 4 -dimethyl-piperazinium iodide (ADMP) and N 1 -phenyl- N 4 -dimethyl-piperazinium iodide (DMPP) with central nicotinic actionBioorganic & Medicinal Chemistry, 1999
- 3-(Piperazinylpropyl)indoles: Selective, Orally Bioavailable h5-HT1DReceptor Agonists as Potential Antimigraine AgentsJournal of Medicinal Chemistry, 1999
- Effect of Modifications of the Alkylpiperazine Moiety of Trazodone on 5HT2Aand α1Receptor Binding AffinityJournal of Medicinal Chemistry, 1999
- Novel Non-Peptide Fibrinogen Receptor Antagonists. 1. Synthesis and Glycoprotein IIb-IIIa Antagonistic Activities of 1,3,4-Trisubstituted 2-Oxopiperazine Derivatives Incorporating Side-Chain Functions of the RGDF PeptideJournal of Medicinal Chemistry, 1998
- A New Palladium-Catalyzed Intramolecular Allylation to Pyrrolidin-2-ones1The Journal of Organic Chemistry, 1998