Single Step Syntheses of ω-9-Fluorenylmethyl Esters of Aspartic and Glutamic Acids
- 1 April 1992
- journal article
- research article
- Published by Taylor & Francis in Synthetic Communications
- Vol. 22 (7) , 1001-1005
- https://doi.org/10.1080/00397919208019289
Abstract
Base lability of the 9-fluorenylmethyl ester makes this group useful in solid phase peptide synthesis when used in combination with the tBoc methodology for preparing cyclic peptides. We describe a simple one step synthesis of the 9-fluorenylmethyl esters of aspartic and glutamic acids.Keywords
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