3D-structure of human estrogenic 17β-HSD1: binding with various steroids
- 30 June 1999
- journal article
- review article
- Published by Elsevier in The Journal of Steroid Biochemistry and Molecular Biology
- Vol. 69 (1-6) , 425-429
- https://doi.org/10.1016/s0960-0760(99)00062-x
Abstract
No abstract availableKeywords
This publication has 13 references indexed in Scilit:
- Synthesis and evaluation of estradiol derivatives with 16α-(bromoalkylamide), 16α-(bromoalkyl) or 16α-(bromoalkynyl) side chain as inhibitors of 17β-hydroxysteroid dehydrogenase type 1 without estrogenic activityBioorganic & Medicinal Chemistry, 1996
- The crystallogenesis of a human estradiol dehydrogenase-substrate complexJournal of Crystal Growth, 1996
- Crystal structure of human estrogenic 17β-hydroxysteroid dehydrogenase complexed with 17β-estradiolNature Structural & Molecular Biology, 1996
- Structure of human estrogenic 17β-hydroxysteroid dehydrogenase at 2.20 å resolutionStructure, 1995
- N-butyl, N-methyl, 11-[3′,17′ β-(dihydroxy)-1′,3′,5′(10′)- estratrien-16′ α-yl]-9(R/S)-bromo undecanamide: synthesis and 17β-HSD inhibiting, estrogenic and antiestrogenic activitiesSteroids, 1994
- Crystallization and Preliminary X-ray Diffraction Analysis of the Complex of Human Placental 17β-Hydroxysteroid Dehydrogenase with NADP+Journal of Molecular Biology, 1993
- Hydrogen bonding in steroidogenesis: Studies on new heterocyclic analogs of estrone that inhibit human estradiol 17β-dehydrogenaseBiochemical and Biophysical Research Communications, 1991
- Trifluoromethylacetylenic alcohols as affinity labels: inactivation of estradiol dehydrogenase by a trifluoromethylacetylenic secoestradiolJournal of Medicinal Chemistry, 1990
- Preparation of 14,15-secoestra-1,3,5(10)-trien-15-ynes, inhibitors of estradiol dehydrogenaseSteroids, 1989
- Human placental estradiol 17.beta.-dehydrogenase: sequence of a histidine-bearing peptide inthe catalytic regionBiochemistry, 1986