Asymmetric Synthesis of Active Pharmaceutical Ingredients

This publication has 272 references indexed in Scilit:

• Developing Processes for Crystallization-Induced Asymmetric Transformation
  Organic Process Research & Development, 2005
• Asymmetry on large scale: the roadmap to stereoselective processes
  Nature Reviews Drug Discovery, 2005
• Chemistry Development of a Convergent Route to Trecetilide Hemi-Fumarate
  Organic Process Research & Development, 2005
• Development of Jacobsen Asymmetric Epoxidation and Sharpless Asymmetric Dihydroxylation Methods for the Large-Scale Preparation of a Chiral Dihydrobenzofuran Epoxide
  Organic Process Research & Development, 2003
• Synthesis of Both Enantiomers of a P-Chirogenic 1,2-Bisphospholanoethane Ligand via Convergent Routes and Application to Rhodium-Catalyzed Asymmetric Hydrogenation of CI-1008 (Pregabalin)
  Journal of the American Chemical Society, 2003
• In Situ Recycling of Chiral Ligand and Surplus Nucleophile for a Noncatalytic Reaction: Amplification of Process Throughput in the Asymmetric Addition Step of Efavirenz (DMP 266)
  Organic Process Research & Development, 2003
• Efficient Synthesis of NK₁ Receptor Antagonist Aprepitant Using a Crystallization-Induced Diastereoselective Transformation
  Journal of the American Chemical Society, 2003
• A simplified procedure for the stereospecific transformation of 1,2-diols into epoxides
  Tetrahedron, 1992
• Asymmetric reduction of 7,8‐difluoro‐3‐methyl‐2H‐1,4‐benzoxazine. Synthesis of a key intermediate of (S)‐(‐)‐ofloxacin (DR‐3355)
  Journal of Heterocyclic Chemistry, 1991
• Asymmetric Catalytic Hydrogenation with an Optically Active Phosphinerhodium Complex in Homogeneous Solution
  Angewandte Chemie International Edition in English, 1968