Palladium-Catalyzed Arylation of Electron-Rich Heterocycles with Aryl Chlorides
Top Cited Papers
- 15 March 2007
- journal article
- letter
- Published by American Chemical Society (ACS) in Organic Letters
- Vol. 9 (8) , 1449-1451
- https://doi.org/10.1021/ol0702324
Abstract
Palladium-catalyzed C−H activation: cheap aryl chlorides can now be used for the arylation of a wide variety of electron-rich heterocycles. The key to the success of this reaction is the use of a bulky, electron-rich phosphine ligand. No copper additives are needed.Keywords
This publication has 24 references indexed in Scilit:
- Regioselective Synthesis of 1,5-Diaryl-1H-imidazoles by Palladium-Catalyzed Direct Arylation of 1-Aryl-1H-imidazolesThe Journal of Organic Chemistry, 2005
- Palladium-Catalyzed Cross-Coupling of Pyrrole Anions with Aryl Chlorides, Bromides, and IodidesOrganic Letters, 2004
- Palladium-Catalyzed Arylation and Heteroarylation of IndolizinesOrganic Letters, 2004
- Palladium-catalyzed direct arylation of thiazoles with aryl bromidesTetrahedron, 2003
- Direct Arylation via Cleavage of Activated and Unactivated C-H BondsPublished by Springer Nature ,2002
- Regioselective Palladium-Catalyzed Arylation of 2-FuraldehydeOrganic Letters, 2001
- Extension of the Heck reaction to the arylation of activated thiophenesJournal of Organometallic Chemistry, 1998
- Palladium-Catalyzed Arylation of Azole Compounds with Aryl Halides in the Presence of Alkali Metal Carbonates and the Use of Copper Iodide in the ReactionBulletin of the Chemical Society of Japan, 1998
- Palladium-catalyzed Cross-coupling Ractions of Chloropyrazines with Aromatic HeterocyclesHETEROCYCLES, 1992
- Palladium-catalyzed Coupling Reaction of Chloropyrazines with IndoleHETEROCYCLES, 1985